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高国锐

作者:宋杰 时间:2024-08-23 浏览量:

姓名:高国锐 

 

说明:E:\DSCN9284.JPG

职称: 

讲师 

专业: 

药物化学 

博(硕)导: 


最终学历: 

博士研究生 

联系电话: 

0531-88233745 

电子邮件: 

gaoguorui2001@163.com 

简历及研究领域 

个人简介: 

研究方向: 

(1)小分子药物化学研究 

(2)药物与精细化学品合成工艺研究 

代表性论文 

5.Guo-Rui Gao, Ling-Hua Meng, Yong-Cong Lv, Su-Feng Cao, Lin-Jiang Tong, Li-Xin Wei, Jian Ding, Hua Xie, Wen-Hu Duan* Design, synthesis and biological evaluation of biphenylurea derivatives as VEGFR-2 kinase inhibitors (II).CHINESE CHEM LETT.2016, 27(2), 200-204

4.Guo-Rui Gao, Ling-Hua Meng, Lin-Jiang Tong, Li-Xin Wei, Jian Ding, Hua Xie, Wen-Hu Duan* Design, synthesis and biological evaluation ofO-linked indoles as VEGFR-2 kinase inhibitors (I).CHINESE CHEM LETT.2015, 26(9), 1165-1168

3.Guo-Rui Gao, Jia-Li Liu, De-Shen Mei, Jian Ding, Ling-Hua Meng, Wen-Hu Duan* Design, synthesis and biological evaluation of acylhydrazone derivatives as PI3K inhibitors.CHINESE CHEM LETT.2015, 26(1), 118-120

2.Liu JL,Gao GR(共同第一), Zhang X, Cao SF, Guo CL, Wang X, Tong LJ, Ding J, Duan WH, Meng LH*. DW09849, a selective phosphatidylinositol 3-kinase (PI3K) inhibitor, prevents PI3K signaling and preferentially inhibits proliferation of cells containing the oncogenic mutation p110alpha (H1047R).J Pharmacol Exp Ther.2014; 348: 432-441

1.替莫西林钠的制备方法.中国专利:CN103910748A

研究课题 



荣誉称号 



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